南方科技大学知识苑(SUSTech KC): Enantioselective Construction of Vicinal Sulfur-functionalized Quaternary and Tertiary Stereocenters via Organocatalytic Michael Addition of 5H-Thiazol-4-ones to 1-Azadienes

题名	Enantioselective Construction of Vicinal Sulfur-functionalized Quaternary and Tertiary Stereocenters via Organocatalytic Michael Addition of 5H-Thiazol-4-ones to 1-Azadienes
作者	Li, Fushuai 1; Zhang, Chen 1; Cheng, Yuyu2 ; Jia, Qianfa 3; Li, Wenjun 1; Liu, Kun 1; Li, Pengfei2,4
通讯作者	Liu, Kun; Li, Pengfei
共同第一作者	Li, Fushuai; Zhang, Chen; Cheng, Yuyu
发表日期	2020-07-17
DOI	10.1002/ajoc.202000272
发表期刊	Asian Journal of Organic Chemistry 影响因子和分区
ISSN	2193-5807
EISSN	2193-5815
卷号	9 期号:8页码:1183-1186
摘要	An organocatalytic enantioselective Michael addition of 5H-thiazol-4-ones to 1-azadienes has been developed. In the presence of chiral phosphoric acid, a series of optically active benzofuran derivatives featured by vicinal sulfur-containing quaternary and tertiary stereocenters were obtained in high yields (71-99%) with high stereoselectivities (70-96%eeand 8 : 1-20 : 1 d.r.).
关键词	Michael Addition 5h-thiazol-4-ones Chiral Phosphoric Acid 1-azadienes
相关链接	[来源记录]
收录类别	SCI
语种	英语
学校署名	通讯
资助项目	National Natural Science Foundation of China[21502043][21871128] ; Special Funds of the Taishan Scholar Program of Shandong Province[tsqn201812047] ; Natural Science Foundation of Shandong Province[ZR2017JL011] ; Shenzhen Innovation of Science and Technology Commission[ZDSYS201802081843490]
WOS研究方向	Chemistry
WOS类目	Chemistry, Organic
WOS记录号	WOS:000548856500001
出版者	WILEY-V C H VERLAG GMBH
来源库	Web of Science
引用统计	被引频次[WOS]：14
成果类型	期刊论文
条目标识符	http://sustech.caswiz.com/handle/2SGJ60CL/141369
专题	理学院_化学系
作者单位	1.Qingdao Univ, Sch Pharm, Dept Med Chem, Qingdao 266021, Shandong, Peoples R China 2.Southern Univ Sci & Technol SUSTech, Coll Sci, Dept Chem, Shenzhen 518055, Guangdong, Peoples R China 3.Yangtze Normal Univ, Coll Chem & Chem Engn, Chongqing Key Lab Inorgan Special Funct Mat, Chongqing 408100, Peoples R China 4.SUSTech, Shenzhen Key Lab Marine Archaea Geoom, Shenzhen, Peoples R China
通讯作者单位	化学系; 南方科技大学
推荐引用方式 GB/T 7714	Li, Fushuai,Zhang, Chen,Cheng, Yuyu,et al. Enantioselective Construction of Vicinal Sulfur-functionalized Quaternary and Tertiary Stereocenters via Organocatalytic Michael Addition of 5H-Thiazol-4-ones to 1-Azadienes[J]. Asian Journal of Organic Chemistry,2020,9(8):1183-1186.
APA	Li, Fushuai.,Zhang, Chen.,Cheng, Yuyu.,Jia, Qianfa.,Li, Wenjun.,...&Li, Pengfei.(2020).Enantioselective Construction of Vicinal Sulfur-functionalized Quaternary and Tertiary Stereocenters via Organocatalytic Michael Addition of 5H-Thiazol-4-ones to 1-Azadienes.Asian Journal of Organic Chemistry,9(8),1183-1186.
MLA	Li, Fushuai,et al."Enantioselective Construction of Vicinal Sulfur-functionalized Quaternary and Tertiary Stereocenters via Organocatalytic Michael Addition of 5H-Thiazol-4-ones to 1-Azadienes".Asian Journal of Organic Chemistry 9.8(2020):1183-1186.